ADENOSINE A2B RECEPTOR AGONIST FOR THE TREATMENT OF MUSCULOSKELETAL CONDITIONS Application EP-3782622-A1 European Patent Office 24 Feb 2021
2-(N-pyrazolo)adenosines with application as adenosine A2A receptor agonists Grant US-RE47351-E1 United States of America 16 Apr 2019
Process for preparing an A2A-adenosine receptor agonist and its polymorphs Grant US-RE47301-E1 United States of America 19 Mar 2019
Anhydrous polymorphs of [(2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-YL)-3,4-dihydroxy… Grant US-9718853-B2 United States of America 01 Aug 2017
Combination, kit and method of reducing intraocular pressure Grant US-9370530-B2 United States of America 21 Jun 2016
Myocardial perfusion imaging methods and compositions Grant US-9289446-B2 United States of America 22 Mar 2016
Method of reducing intraocular pressure in humans Grant US-9289383-B2 United States of America 22 Mar 2016
Anhydrous polymorphs of [(2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy… Grant US-9278991-B2 United States of America 08 Mar 2016
Substituted dicyanopyridines and use thereof Grant US-9187428-B2 United States of America 17 Nov 2015
Substituted aryloxazoles and their use Application US-9095582-B2 United States of America 04 Aug 2015
Process for preparing an A2A-adenosine receptor agonist and its polymorphs Grant US-9085601-B2 United States of America 21 Jul 2015
Adenosine A1 agonists for the treatment of glaucoma and ocular hypertension Application US-9040566-B2 United States of America 26 May 2015
Myocardial perfusion imaging methods and compositions Grant US-8906878-B2 United States of America 09 Dec 2014
2-alkoxy-substituted dicyanopyridines and their use Application US-8791146-B2 United States of America 29 Jul 2014
Alkylamino-substituted dicyanopyridines and their amino acid ester prodrugs Application EP-2743270-A1 European Patent Office 18 Jun 2014
Dipeptoid prodrugs and the use thereof Application US-8703696-B2 United States of America 22 Apr 2014
Substituted 4-amino-3,5-dicyano-2-thiopyridines and use thereof Grant US-8703934-B2 United States of America 22 Apr 2014
Substituted bipyridine derivatives and their use as adenosine receptor ligands Grant US-8653109-B2 United States of America 18 Feb 2014
Purine derivatives as adenosine A1 receptor agonists and methods of use thereof Grant US-8609833-B2 United States of America 17 Dec 2013
Substituted azabicyclic compounds and the use thereof Grant US-8609686-B2 United States of America 17 Dec 2013
Monohydrate of (1-{9-[4S,2R,3R,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-6-aminopurin… Grant US-8524883-B2 United States of America 03 Sep 2013
Myocardial perfusion imaging methods and compositions Grant US-8470801-B2 United States of America 25 Jun 2013
Heteroaryl-substituted dicyanopyridines and their use Grant US-8426602-B2 United States of America 23 Apr 2013
Alkylamino-substituted dicyanopyridines and their amino acid ester prodrugs Application US-8420825-B2 United States of America 16 Apr 2013
3-cyano 5-thiazaheteroaryl-dihydropyridine and the use thereof for the treatment of… Grant US-8404723-B2 United States of America 26 Mar 2013
3,4-Dihydro-4-oxo-5-aryl-pyrido[2,3-d]pyrimidine-6-carbonitriles as Adenosin Receptor… Application EP-2556831-A1 European Patent Office 13 Feb 2013
6-Cyano-substituted Pyrido[2,3-d]pyrimidines as Adenosin Rezeptor Ligands for the… Application EP-2556856-A1 European Patent Office 13 Feb 2013
Cyclically substituted 3,5-dicyano-2-thiopyridines and use thereof Grant US-8304412-B2 United States of America 06 Nov 2012
Process for preparing an A2A-adenosine receptor agonist and its polymorphs Grant US-8268988-B2 United States of America 18 Sep 2012
Substituted 2, 6-diamino-3, 5-dicyano-4-arylpyridines and their use as adenosine-receptor-s… Grant US-8242281-B2 United States of America 14 Aug 2012
Purine derivatives as adenosine A1 receptor agonists and methods of use thereof Grant US-8183224-B2 United States of America 22 May 2012
Myocardial perfusion imaging methods and compositions Grant US-8133879-B2 United States of America 13 Mar 2012
Purine derivatives and methods of use thereof Grant US-8133880-B2 United States of America 13 Mar 2012
Process for preparing an A2A-adenosine receptor agonist and its polymorphs Grant US-8106183-B2 United States of America 31 Jan 2012
SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF Application WO-2012000945-A1 World Intellectual Property Organisation (WIPO) 05 Jan 2012
Process for preparing an A2A-adenosine receptor agonist and its polymorphs Grant US-7956179-B2 United States of America 07 Jun 2011
INTRATHECAL TREATMENT OF NEUROPATHIC PAIN WITH A2AR AGONISTS Application EP-2240020-A4 European Patent Office 11 May 2011
Purine Derivatives and methods of use thereof Grant US-7863253-B2 United States of America 04 Jan 2011
INTRATHECAL TREATMENT OF NEUROPATHIC PAIN WITH A2AR AGONISTS Application EP-2240020-A1 European Patent Office 20 Oct 2010
Alkylamino-substituted dicyanopyridines and their amino acid ester prodrugs Application DE-102009006602-A1 Germany 05 Aug 2010
ALKYLAMINE-SUBSTITUTED DICYANOPYRIDINE AND AMINO ACID ESTER PRODRUGS THEREOF Application WO-2010086101-A1 World Intellectual Property Organisation (WIPO) 05 Aug 2010
Purine derivatives and methods of use thereof Grant US-7732424-B2 United States of America 08 Jun 2010
Azabicyclic-substituted 5-aminopyrazoles and their use Application DE-102008039082-A1 Germany 25 Feb 2010
Heteroaryl-substituted dicyanopyridines and their use Application DE-102008013587-A1 Germany 17 Sep 2009
Cycloalkoxy-substituted 4-phenyl-3,5-dicyanopyridines and their use Application DE-102008008838-A1 Germany 20 Aug 2009
FUSED CYNOPRYRIDINES AND THE USE THEREOF Application WO-2009080198-A1 World Intellectual Property Organisation (WIPO) 02 Jul 2009
Purine Derivatives as adenosine A1 receptor agonists and methods of use thereof Grant US-7423144-B2 United States of America 09 Sep 2008
8-heteroaryl xanthine adenosine A2B receptor antagonists Grant US-7335655-B2 United States of America 26 Feb 2008
8-Heteroaryl xanthine adenosine A2B receptor antagonists Grant US-7205403-B2 United States of America 17 Apr 2007
Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof Grant US-7135486-B1 United States of America 14 Nov 2006
Substituted 2-carba-3,5-dicyano-4-aryl-6-aminopyridines and the use of the same as… Grant US-7129255-B2 United States of America 31 Oct 2006
Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding… Grant US-7078417-B2 United States of America 18 Jul 2006
Substituted 2-thio-3, 5-dicyano-4-phenyl-6-aminopyridines and their use as adenosine… Grant US-7045631-B2 United States of America 16 May 2006
Method for identifying and using A2B adenosine receptor antagonists to mediate mammalian… Application US-6894021-B2 United States of America 17 May 2005
Methods for reducing intraocular pressure using A3 adenosine receptor antagonists Grant US-6528516-B1 United States of America 04 Mar 2003