Cyclopropyl dihydroquinoline sulfonamide compounds Grant US-11807634-B2 United States of America 07 Nov 2023
Composition and methods for treating intestinal hyperpermeability Grant US-11786496-B2 United States of America 17 Oct 2023
Compositions and methods for treating autism Grant US-11633372-B2 United States of America 25 Apr 2023
Combinations comprising positive allosteric modulators or orthosteric agonists of… Grant US-11369606-B2 United States of America 28 Jun 2022
Combinations comprising positive allosteric modulators or orthosteric agonists of… Grant US-11103506-B2 United States of America 31 Aug 2021
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyridinyl-2′-ones Grant US-11071729-B2 United States of America 27 Jul 2021
Tyrosine derivatives and compositions comprising them Grant US-11058638-B2 United States of America 13 Jul 2021
Compositions and methods for treating intestinal hyperpermeability Grant US-10857118-B2 United States of America 08 Dec 2020
Compositions and methods for treating autism Grant US-10813901-B2 United States of America 27 Oct 2020
Compositions and methods for treating autism Grant US-10751313-B2 United States of America 25 Aug 2020
Alkynyl dihydroquinoline sulfonamide compounds Grant US-10729684-B2 United States of America 04 Aug 2020
Substituted 6,7-dihydropyrazolo[1,5-a]pyrazines as negative allosteric modulators of… Grant US-10584129-B2 United States of America 10 Mar 2020
Combinations comprising positive allosteric modulators or orthosteric agonists of… Grant US-10537573-B2 United States of America 21 Jan 2020
Compositions and methods for treating intestinal hyperpermeability Application US-10517845-B2 United States of America 31 Dec 2019
Bicyclic ketone sulfonamide compounds Application US-10472356-B2 United States of America 12 Nov 2019
Pharmaceutical Compositions And Methods Application US-20190275117-A1 United States of America 12 Sep 2019
Alkyl dihydroquinoline sulfonamide compounds Application US-10383866-B2 United States of America 20 Aug 2019
PHARMACEUTICAL COMPOSITIONS AND METHODS Application US-20190201378-A1 United States of America 04 Jul 2019
Pharmaceutical compositions and methods Application US-10307465-B2 United States of America 04 Jun 2019
Pharmaceutical compositions and methods Application US-10272068-B2 United States of America 30 Apr 2019
Substituted 6,7-dihydropyrazolo[1,5-a]pyrazines as negative allosteric modulators of… Grant US-10106542-B2 United States of America 23 Oct 2018
Compositions and methods for treating intestinal hyperpermeability Application US-10085959-B2 United States of America 02 Oct 2018
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of… Grant US-10071095-B2 United States of America 11 Sep 2018
Pharmaceutical compositions and methods Application US-10010590-B2 United States of America 03 Jul 2018
Pharmaceutical compositions and methods Application US-9895425-B2 United States of America 20 Feb 2018
Compositions and methods for treating intestinal hyperpermeability Application US-9763903-B2 United States of America 19 Sep 2017
Composition and methods for treating intestinal hyperpermeability Application US-9757348-B2 United States of America 12 Sep 2017
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention… Grant US-9737533-B2 United States of America 22 Aug 2017
1,2,4-triazolo[4,3-a]pyridine compounds and their use as positive allosteric modulators… Grant US-9708315-B2 United States of America 18 Jul 2017
Tyrosine derivatives and compositions comprising them Application US-9585841-B2 United States of America 07 Mar 2017
PHARMACEUTICAL COMPOSITIONS AND METHODS Application US-20160263198-A1 United States of America 15 Sep 2016
PHARMACEUTICAL COMPOSITIONS AND METHODS Application US-20160263149-A1 United States of America 15 Sep 2016
Compositions and methods for treating intestinal hyperpermeability Application US-9326962-B2 United States of America 03 May 2016
Compositions and methods for treating intestinal hyperpermeability Application US-9308188-B2 United States of America 12 Apr 2016
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators… Grant US-9271967-B2 United States of America 01 Mar 2016
1, 4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric… Grant US-9266834-B2 United States of America 23 Feb 2016
1,2,4-triazolo [4,3-a] pyridine derivatives and their use for the treatment of prevention… Grant US-9226930-B2 United States of America 05 Jan 2016
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyridinyl-2′-ones Grant US-9132122-B2 United States of America 15 Sep 2015
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones Grant US-9114138-B2 United States of America 25 Aug 2015
7-aryl-1,2,4-triazolo[4,3-A]pyridine derivatives and their use as positive allosteric… Grant US-9085577-B2 United States of America 21 Jul 2015
1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric… Grant US-9067891-B2 United States of America 30 Jun 2015
Bicyclic aryl and heteroaryl sodium channel inhibitors Application US-9012443-B2 United States of America 21 Apr 2015
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators… Grant US-9012448-B2 United States of America 21 Apr 2015
1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric… Grant US-8993591-B2 United States of America 31 Mar 2015
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators… Grant US-8946205-B2 United States of America 03 Feb 2015
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention… Grant US-8937060-B2 United States of America 20 Jan 2015
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives Grant US-8906939-B2 United States of America 09 Dec 2014
1, 4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric… Grant US-8841323-B2 United States of America 23 Sep 2014
Imidazo[1,2-A]pyridine derivatives and their use as positive allosteric modulators of… Grant US-8785486-B2 United States of America 22 Jul 2014
1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones Grant US-8748621-B2 United States of America 10 Jun 2014
1,3-disubstituted-4-phenyl-1H-pyridin-2-ones Grant US-8722894-B2 United States of America 13 May 2014
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric… Grant US-8716480-B2 United States of America 06 May 2014
Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors Grant US-8697689-B2 United States of America 15 Apr 2014
3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors Grant US-8691849-B2 United States of America 08 Apr 2014
Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors Grant US-8691813-B2 United States of America 08 Apr 2014
PHARMACEUTICAL COMPOSITIONS AND METHODS Application US-20130184214-A1 United States of America 18 Jul 2013
Pharmaceutical compositions and methods Application US-8481498-B1 United States of America 09 Jul 2013
COFERONS AND METHODS OF MAKING AND USING THEM Application WO-2009126290-A2 World Intellectual Property Organisation (WIPO) 15 Oct 2009